Yagman said:Yeah, I guess you'll just have to let this one play out. I just happen to know how it ends.
Bobo said:Funny, if PA made that claim and was banned, all hell would break loose with his little fanclub. If anyone else did it, they would deserve it.
Bobo said:Invalid Link Removed
:lol:
NoSwtTea4U said:So back to the Topic of the Thread :rant: ....
Buc4Life04 said:Then people even admit they got banned from here and come back.
So AM has to be doing something right.
\/ \/ \/ \/ HAHAHA Good one BObo
Glad to see I was not the only one who found this timing a bit suspect.TheOMEGA said:the straw on the camels back for me is how he tested DS stuff then right after the expose' he comes out with ATD.....
Author L. Rea said:It seems that the first analog we will be focusing on is 4,17b-diydroxyestra-4,9,11-trien-3-one. Not that some of the others do not hold interest both from a research and potential point, but simply because we have already moved so far ahead on this one and one other...but the vote is in.
Thank you lads. I appreciate your time and interests.
And Bruce, thank you for sharing yours with us!
I see this as a THP ether. Thoughts?
Bobo said:Dr.D,
Please take this stuff to email.
SJA said:I guess DrD should be posting that in his own forum?
SJA said:You police it well and we've had a thread discussing this and thanking you. You never worried about what others would say about you if you banned someone....why start now?
As for the other points I made aobut banning, I was being more sarcastic than anything. Policies won't change here because of public opinion.
thanks, it was/ is an uncomfortable event that has been stumbled on, but when someone is like that its hard not to say anything about itBobo said:You hit the nail on the head. On that note, I'm off to bed. Finally someone who see's it for what it is.
...except size
Man...They actually think this guy is sincere. The flock continues to grow...LOL....
Is this the same BK?BKneller said:Matt Cahill is toast! I am going to litigate against DS too. I'm not going into specifics but lets just say I have a
better than average case against him IMHO (as well as the other cloners).
So yeah, I plan to sue Designer Supps for selling ATD if they are still selling it after my application for ATD is published
by the USPTO.
BK
Its sad to see this complete change of behaviour 2 months after.Invalid Link Removed
Matt and I will work this out so that no matter what, both of us end upwith an effective anti-aromatase based on ATD to sell. I am not looking to screw him or anyone else. He's a pretty nice guy, smart too. So let Matt/me/lawyers work something out. In the mean time, he is gonna continue to sell Rebound XT and Gaspari will sell Novedex XT.
This is fair for the time being until we work this out between us.
BK
DR.D said:Author,
I am not sure why you hooked up with BK and it is not my style to judge. Plus, it is beyond the scope of the my point. Therefore, although he has threatened litigation against my company, I still respect you and would like to see you advance. 4-subs are tricky, I have been looking to exploit one too, but I really can't recommend any of your choices. I'm not even sure if #4 is chemically possible/stable. So while I may not be the "best chemist in China..." I could probably still help you not waste any more money than necessary. Like I have told you previously, I think we have much more to gain from one another working together than at odds with one another. The patent app won't stick in court, we both know why, and it's stupid to bluff one anther and promote all this drama. At the risk of sounding chauvinistic, let's leave that to women and soap operas! You never know when the government may choose to put us all out of work. Why fight one another and talk about legal action? I know that we are technically rivals, but it's still counter productive and does not advance the science or the sport. This is a huge waste of time when we need to be moving ahead and developing new compounds as fast as possible. Feel free to PM or hushmail me and I will explain my view on hetero sub's on the 4 carbon, only if you like. Otherwise, please forgive me posting on your thread and I will stay away from this one in the future.
Best of luck with that. I have been polite(as always) but I can't say the same for him.TheOMEGA said:hope he aplogizes as well for some of the things he has said as well
I'm not a huge PA fan but he has nothing to apologize to you for.TheOMEGA said:in the spirit of good will and forgiveness I am sorry to PA for soem of the things I said in anger
hope he aplogizes as well for some of the things he has said as well
LCSULLA said:Doc, can you tell us which compounds Mr. Rea listed do you think will be "workable" And do you think the THP ether will be viable?
Author L. Rea said:It seems that the first analog we will be focusing on is 4,17b-diydroxyestra-4,9,11-trien-3-one. Not that some of the others do not hold interest both from a research and potential point, but simply because we have already moved so far ahead on this one and one other...but the vote is in.
Thank you lads. I appreciate your time and interests.
And Bruce, thank you for sharing yours with us!
I see this as a THP ether. Thoughts?
Bobo said:Hey Bruce,
Its very simple. If you want to remain here you don't bash a sponsor. I'm not going to put up with it. THis is your last warning. Quit the BS or you will be gone just like PA. Time to keep you business to yourself. Let this be the last time we have any problems.
Both directions? :think:BKneller said:Noted. Will comply Bobo.
Fair enough? I also trust this goes in both directions then.
BK
DR.D said:OK, you asked for it!
1) 4,17b-diydroxyestra-4,9,11-trien-3-one
2) 17a-methyl-4-hydroxy-4,9-dien-3-one
3) 17a-methyl-2-hydroxymethylene-4-hydroxy-5-androstan-3-one
4) 4-hydroxy-1-methyl-5a-androst-1-en-3-one
5) 4-hydroxy-17a-methyl-2-oxa-5a-androstane-3-one
6) 4-hydroxy-17a-methyl-androsta-1,4-dien-3-one
The 4 sub has advantages. First it creates a hormone that can not aromatize. Also, it acts as a 5-reductase inhibitor. So you won't form estrogen or DHT with this these type compounds. There are 3 mains groups that convey signifigant activity at the 4 position: halogens, hydroxyl, and the methyl. The main issues with these compounds are the added resonance of the 3, 4 & 5 functions. 4-carbon subs also reduce polarity of the 3-one. You know what, screw the outline, this will take forever. I'll tell you like this.. Compound#1: Why? Why make a designer androgen that already won't aromatize non-aromatizable? The oral bioavailability may be better that one would guess, but I suspect the intrinsic potency would be lacking. Start with an aromatizable compound most likely. #2: I'm not sure what this is, a C-19 steroid? Part of the compound name seems to be missing, it's impossible to say what the skeleton is, but it has the same issues as the first reguardless. The improved electron delocalization of the diene and triene systems convey stability, but the 4 sub would weaken it over the original parent compound. #3: Severe steric distortion of the A & B ring conjuctions throwing the face out of plane, I don't even think humans have a receptor that would accommodate that molecule! This structure could possess 4 different sterioisomers (just considering the A-ring) so it would be naturally weak as the racemic mixture. #4: Same issue as the first one and it is also unstable. The charge on the 5 carbon would likely be negative. 4 subs generally need a 4-ene system. The 3 carbon may also adopt a positive charge stretching the 3-one bond. 4-ene protects 3=O, as both have shorter bond lengths. #5: This one may have activity but it would be very low I'd guess. Also, it has the same issue as the first one. Why not choose an aromatizable base to begin with when looking at this issue? It defeats the main purpose of the 4-OH! #6: This compound may possess activity too, but the same issues apply as the third. Because the carbonyl bond is stretched longer than usual with a 4 hetero sub, you may have a compound with equilibrated resonance to give the effect of non-aromatizable dbol. Also the planarity of the 1,4-ene system would be skewed which kills the real beauty of dbol. The potency may be as much as 50% that of dbol itself. It's hard to guess. To summarize, this is a hard area to exploit and you need more than just a hunch to do it successfully. Or, you need lots of money and after you prep 100 compounds, you may by luck finally run across one! Or who know, I may be totally wrong and all 6 of these are the strongest hormones ever invented!! But if Matt told me he wanted another 4 carbon modified supp, I would have a different choice, maybe a 4-methyl. There may only be about 2 or 3 more good compounds in this series yet to be discovered. The THP ether would be viable with 1, 5 & 6. If I had to choose one of these, I'd go with the 17-ether of 6.
cool I was looking forward to your input hereBKneller said:Noted. Will comply Bobo.
Fair enough
TheOMEGA said:cool I was looking forward to your input here![]()
LCSULLA said:BK,
Can you tell us about 2 and 3?
While my judgement on Prostan is suspended (its only been one week), I completely agree on BK on this. We dont need more methyls, no matter how strong they are.BKneller said:As an aside...I don't know why so many people think that you must "alpha alkylate at C-17a" to have an effective oral. The feedback on our stanozolol analog has been FANTASTIC do date and this is a "non-methyl" - it seems to be 50% less potent than "regular stanozolol" but so what? Our version won't get you a date with the local district attorney
While we (Author and I) do plan on launching a few C-17a modified compounds in the future (you think we have discussed EVERYTHING here? Not a chance!) we both agree that there is a much larger market for people who want a 'safer kinder, proto-steroid' so to speak and for people who want 'something to stack with a methyl' that may already be available to them.
Syr said:While my judgement on Prostan is suspended (its only been one week), I completely agree on BK on this. We dont need more methyls, no matter how strong they are.
We could need some in the future, but only if they prove to be safe on liver and lipid like only m4ohn was.
There are 2 (soon 3) strong methyl bulkers on the market already and people need something to stack with them to tailor more advanced cycles.
BTW, I encourage for an accurate and extensive (n>5) alpha-testing of erverything and a sound dosing protocol. Not every thp ether must be dosed at 25mgx3
cheers
[edit: ester for ether]
BKneller said:Noted. Will comply Bobo.
Fair enough? I also trust this goes in both directions then.
BK
BKneller said:I have a BS degree in Clinical Laboratory Science and a BS degree in Nursing. I hold registration/certification/licensure in both disciplines.
I spent 3 years in pharmacy school before switching majors to Lab Science so I have all the basic undergrad chem/physics/bio course and a few other unique ones. I have 3 graduate course under my belt (I am not pursuing a grad degree at this time).
I never claimed to be a degreed chemist either. Just a guy with an insight for creating useful stuff.
Dr. D:DR.D said:Author,
I am not sure why you hooked up with BK and it is not my style to judge. Plus, it is beyond the scope of the my point. Therefore, although he has threatened litigation against my company, I still respect you and would like to see you advance. 4-subs are tricky, I have been looking to exploit one too, but I really can't recommend any of your choices. I'm not even sure if #4 is chemically possible/stable. So while I may not be the "best chemist in China..." I could probably still help you not waste any more money than necessary. Like I have told you previously, I think we have much more to gain from one another working together than at odds with one another. The patent app won't stick in court, we both know why, and it's stupid to bluff one anther and promote all this drama. At the risk of sounding chauvinistic, let's leave that to women and soap operas! You never know when the government may choose to put us all out of work. Why fight one another and talk about legal action? I know that we are technically rivals, but it's still counter productive and does not advance the science or the sport. This is a huge waste of time when we need to be moving ahead and developing new compounds as fast as possible. Feel free to PM or hushmail me and I will explain my view on hetero sub's on the 4 carbon, only if you like. Otherwise, please forgive me posting on your thread and I will stay away from this one in the future.
Nice, upstanding post AuthorAuthor L. Rea said:Dr. D:
First it seems I owe you and everyone at DS an apology. I realize the words were not mine, but they were said by a good friend of mine, on my forum space, so it is my loss of honor first. I do not support ANYONE attaching another company on my forum or otherwise. It is exactly why I have never posted much. If there are legal issues between company's then that should be left to the lawyers and handled in private. Anything else just destroys the industry and I personally feel that we really do need more companies that will work together. I believe that I have openly supported Matt and you both for your work and products, and certainly will continue to do so (I do not find it likely that DS will start making trash products anytime soon...or in the future). I hope you and Matt will accept my apology, though I would understand if not. Trust is such a rare and precious thing, and like honor, it should be given to those who hold it as part of their soul. Not going estrogenic here, just a fact. And by the way, I do not believe we are rivals, more like lads who have a rare passion for the same industry. You are always welcomed here or anywhere I am.
Bobo and Size:
I want to apologize to both of you as well. My intent was, and still is, to bring some of the brightest lads who think outside the envelope to share with others I respect such as Dr. D. here on the AM board. I am normally not one to openly discuss anything with anyone publicly as it seems that those who think outside the envelope are so often ridiculed for innovation (have any of our products yet failed to set new levels of expectation? The **** works...though many say they won't) until they are copied for gain. But I do enjoy posting here on AM when I have time due to the lack of flamers and childish behavior...for the most part. (Yes, I know I had a temper tantrum a month or so ago...my error)
Bruce is of course, his own man and I never attempt to tell anyone what I feel they should do. Naturally I fully understand and support his or anyone's right to defend their investments where it applies, but not on the AM board, please. I will ask him to continue to share his amazingly passion for products and designs (I have enjoyed many late night discussions with him that bent even my "outside the box" outlooks) as I believe many are interested in what is possible and those who willing to search for it. He is very bright and his passions do run rather deep in ways that would surprise many that only know his temper. It is your board, your call Lads. I just visit because I like the people.
Author L. Rea
PS: Dr. D. I do not have your hushmail addy. Please send it to Raven when you have a minute.