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Boladrol The Side Effects Log
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INFORMATION SECTION
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Boladrol - A Brand New PH from IBE!
--------------------------------------------------------------------------------
Yes, you heard it right! IBE is releasing a new PH to the market.
We have had many great products in the past, but there is nothing and has never been anything offered quite like Boladrol. The potential for this compound is outstanding and a perfect bulking agent for the upcoming winter. This is a very wet compound that will require PCT and is strongly recommended to stack with a good cycle support product.
The new product Boladrol is 7, 17-alpha-dimethyl-androsten-3, 17-diol (Boladiol), the diol version of the steroid Bolasterone.
60 caps, 2mg per cap, Ready in 2-3 weeks!
Bolasterone is the 7, 17 dimethylated version of testosterone and has the reputation as being one of the most potent steroids ever sold. Bolasterone has an anabolic to androgenic ratio that shows it to be 6x more anabolic than methyltestosterone and 3x as androgenic.
Boladrol will be best compared to Anadrol if not stronger. This PH only requires a few milligrams to see strong anabolic and androgenic effects which we were very excited to see first hand during our alpha testing of this compound. Users have been reported to gain up to a pound a day but also not coming off as quick as reported with Anadrol gains.
projected 2-3 week release date of Bolodrol to the public.
--------------------------------
MY OWN PERSONAL NOTES
--------------------------------
WRITTEN BY anthony roberts
Bolasterone (aka Myagen) is simply DiMethyltestosterone (7α,17α-Dimethyltestosterone), or Methyltestosterone (testosterone with a methyl group at the 17th position) but with an additional methyl group (hence “dimethyl”) at the C7 position. The first methyl group (at the 17th position) allows the steroid to pass through the liver and remain active in the blood. The Second methyl group (at the 7th position) prevents it from binding freely to Sex Hormone Binding Globulin (SHBG), thereby allowing much of it to remain unbound and in an active state, and therefore greatly increasing its potency. I think any further comparison to Methyltestosterone (except perhaps with regards to hepatoxicity – the fancy word for liver toxicity) wouldn’t really be warranted.
Chemically, this stuff is closer to Cheque Drops (Mibolerone) than anything else I can think of. Check out their names side-by-side:
•17beta-Hydroxy-7alpha, 17dimethylestr-4-an-3-one (Cheque Drops)
•17beta-Hydroxy-7alpha, 17dimethylandrost-4-an-3-one (Bolasterone)
The difference here, going by the names, is that one is derived from Nandrolone, and the other is derived from Testosterone (Bolasterone). And if we’re interested in a paint-by-numbers account of thses two compounds, Cheque Drops have an anabolic/androgenic ratio of 590:250, while Bolasterone has a 575:300. Clearly they are very, very, similar. This could end up being a nightmare of liver toxic, side-effect producing garbage. On the other hand, maybe it’ll be the greatest stuff ever.
I’m optimistic, personally, and if I had some on hand, I’d try it. So, for what it’s worth, I feel comfortable enough with the compound to not only warrant talking about it, but also to take it personally.
Unfortunately, most of what we (or at least I) know about Bolasterone is really speculative and/or academic. To my knowledge, it wasn’t available anywhere when I wrote my first book, although I noted that its high anabolic rating (575!) would make it a likely candidate to appear on the black market after my book was published. I was right, and DL Pharmaceuticals eventually produced it in limited quantities in 2007, only to disappear again by 2008. Recently, Geneza Pharmaceuticals has put it back on the market, as a 50mg tablet. I can understand why they’d think it would be appealing to anabolic steroid users - it’s 3x as androgenic as testosterone and almost 6x as anabolic! While I realize that those numbers don’t always paint an accurate picture of a steroid’s potency (Halotestin is over 19x as anabolic as testosterone, and it’s virtually useless for muscle gain). (*Note: I don’t work for Geneza Pharmaceuticals, aka Naps/NapsGear, nor any of their competitors.)
Taking a look at the metabolites, none are immediately aromatized into estrogen, but what I’m seeing here is a removal of the 4-5 double bond and the addition of a hydrogen, thereby showing the potential of this steroid to become 5a-reduced version of its former self, or a dihydrodimethyltestosterone. Last time I checked, William Llewellyn had been saying that Bolasterone probably wasn’t able to be 5a-reduced, and likely converts to a highly potent estrogen, but I think the chart on the left clearly shows the opposite. I mention this because even though I think he’s a complete D-Bag, I don’t discount his steroid knowledge. None of the metabolites appear to be aromatized, as the signature alternating double bonds in the A-ring are not apparent at this stage. Is there further metabolism of these metabolites downstream? Are they substrates for something I haven’t examined? I don’t know. Maybe there is. Maybe they are. I have no idea.
Methyltestosterone happens to convert to a very potent form of estrogen, so this might be the case here as well, and Bolasterone may well end up being the kind of stuff we see people finding use to necessarily be in conjunction with an anti-estrogen, like Anastrozole (Arimidex) or Aromasin (Exemestane). Maybe it converts to the frightening 7α,17α-dimethylestradiol. And since Cheque drops are a liver-toxic nightmare, in terms of estrogen-like symptoms, we may see that here too…perhaps similarly to what is seen with Anadrol, which is 5a-reduced and doesn’t convert to estrogen – yet for some reason exhibits estrogen like side effects such as gynecomastia. Hell…maybe we won’t see any conversion to anything, and a ton of side effects anyway (again, Anadrol comes to mind). On the other hand, this stuff is definitely going to be liver toxic. But as for side effects? We may see none.
Then again, perhaps is doesn’t convert to estrogen at all. If Bolasterone undergoes 5a-reduction immediately in the first stage of metabolism, then aromatization would be impossible. On the other hand, if this chart is incomplete, then maybe it does undergo conversion to estrogen.
One thing is for sure: Since Geneza Pharmaceuticals has brought this stuff back into circulation, we’ll find out soon enough.
--------------------------------------------------------------------------------------------
Bolasterone is an oral anabolic steroid which is structurally related to methyltestosterone. It differs only by the addition of a methyl group, which is the reasoning for its chemical name. The addition of this methyl group makes the activity of this steroid far different than its cousin however, and makes any comparison between the two difficult. This drug was first developed in the late 1950’s. It was closely evaluated for anabolic and androgenic effect around 3 years later. The drug was developed by the pharmaceutical company UpJohn, and was sold in the United States during the 1960s under the brand name of Myagen. It was mainly prescribed for the treatment of advanced breast cancer in women, but was also investigated for use on lean tissue sparing activity. The medical use of this drug didn’t last long however, and it soon disappeared off the market not too long after it was released. By the 1980s, the drug had pretty much been forgotten by bodybuilders and athletes. Although bolasterone is no longer produced, the drug remains listed in the U.S Pharmacopeias, suggesting that it wouldn’t be impossible to see the drug available once again as a prescription medication in the U.S, however this remains very unlikely.
Bolasterone is a fairly potent anabolic steroid, measured in human subjects to have approximately twice the anabolic effect of methandrostenolone. Despite being a derivative of testosterone, bolasterone is considerably more anabolic than it is androgenic in nature. Bodybuilders and athletes would often use this drug in bulking cycle, where adding extra weight wasn’t a concern. Bolasterone is a very estrogenic steroid by nature, and one can expect to see all of the common estrogen related side effects when taking this drug, especially in higher doses. Estrogen related side effects can include such things as increased water and fat retention and gyno (the development of unattractive and sometimes painful female breast tissue under the nipples in males). To combat such issues, users often prefer to run some sort of anti estrogen compound such as arimidex or aromasin during cycle. This steroid can also be androgenic and can produce androgen related side effects as well. These side effects can include such things as oily skin, acne, and increased body and facial hair. In women, androgen can cause masculizing side effects such as deepening of the voice, the growth facial hair, and clitoral enlargement. Bolasterone is a C17aa compound, which means that it can be toxic to liver if taken in doses too large or for periods too long. Because of this, users are urged to try to keep cycles under 8 weeks and to run some sort of liver protection product such as liv-52. Like all anabolic steroids, bolasterone will shut down the body’s natural testosterone production, making a post cycle therapy protocol necessary after the drug’s use has been discontinued. Users often choose to run compounds such as clomid and HCG to get the body to start producing testosterone naturally again.
Clinical studies have demonstrated that significant nitrogen retention and weight gain can be induced with a daily dosage of 1-2mg per day. In the case of bodybuilders and athletes looking for performance enhancement purposes, users often choose run a dosage of 2-5mg per day for a period of 6-8 weeks. This level is sufficient for strong increases in muscle size and strength, although such gains will likely be accompanied by significant water retention due to estrogen. Bolasterone is generally not recommended for women due to its very strong nature and tendacy to produce virilizing side effects.
MY NOTES CONTINUE PLEASE READ ON
I'll be back later on tonight to update this page with a flood of information and items to think about regarding this supplement.However in the meantime I will simply leave this sexy piece of eye candy here for all to enjoy.
[/URL][/IMG]
MY NOTES CONTINUE PLEASE READ ON
-----------------------------
INFORMATION SECTION
-----------------------------
Boladrol - A Brand New PH from IBE!
--------------------------------------------------------------------------------
Yes, you heard it right! IBE is releasing a new PH to the market.
We have had many great products in the past, but there is nothing and has never been anything offered quite like Boladrol. The potential for this compound is outstanding and a perfect bulking agent for the upcoming winter. This is a very wet compound that will require PCT and is strongly recommended to stack with a good cycle support product.
The new product Boladrol is 7, 17-alpha-dimethyl-androsten-3, 17-diol (Boladiol), the diol version of the steroid Bolasterone.
60 caps, 2mg per cap, Ready in 2-3 weeks!
Bolasterone is the 7, 17 dimethylated version of testosterone and has the reputation as being one of the most potent steroids ever sold. Bolasterone has an anabolic to androgenic ratio that shows it to be 6x more anabolic than methyltestosterone and 3x as androgenic.
Boladrol will be best compared to Anadrol if not stronger. This PH only requires a few milligrams to see strong anabolic and androgenic effects which we were very excited to see first hand during our alpha testing of this compound. Users have been reported to gain up to a pound a day but also not coming off as quick as reported with Anadrol gains.
projected 2-3 week release date of Bolodrol to the public.
--------------------------------
MY OWN PERSONAL NOTES
--------------------------------
----------------------------------------------------------------------------------------
WRITTEN BY anthony roberts
Bolasterone (aka Myagen) is simply DiMethyltestosterone (7α,17α-Dimethyltestosterone), or Methyltestosterone (testosterone with a methyl group at the 17th position) but with an additional methyl group (hence “dimethyl”) at the C7 position. The first methyl group (at the 17th position) allows the steroid to pass through the liver and remain active in the blood. The Second methyl group (at the 7th position) prevents it from binding freely to Sex Hormone Binding Globulin (SHBG), thereby allowing much of it to remain unbound and in an active state, and therefore greatly increasing its potency. I think any further comparison to Methyltestosterone (except perhaps with regards to hepatoxicity – the fancy word for liver toxicity) wouldn’t really be warranted.
Chemically, this stuff is closer to Cheque Drops (Mibolerone) than anything else I can think of. Check out their names side-by-side:
•17beta-Hydroxy-7alpha, 17dimethylestr-4-an-3-one (Cheque Drops)
•17beta-Hydroxy-7alpha, 17dimethylandrost-4-an-3-one (Bolasterone)
The difference here, going by the names, is that one is derived from Nandrolone, and the other is derived from Testosterone (Bolasterone). And if we’re interested in a paint-by-numbers account of thses two compounds, Cheque Drops have an anabolic/androgenic ratio of 590:250, while Bolasterone has a 575:300. Clearly they are very, very, similar. This could end up being a nightmare of liver toxic, side-effect producing garbage. On the other hand, maybe it’ll be the greatest stuff ever.
I’m optimistic, personally, and if I had some on hand, I’d try it. So, for what it’s worth, I feel comfortable enough with the compound to not only warrant talking about it, but also to take it personally.
Unfortunately, most of what we (or at least I) know about Bolasterone is really speculative and/or academic. To my knowledge, it wasn’t available anywhere when I wrote my first book, although I noted that its high anabolic rating (575!) would make it a likely candidate to appear on the black market after my book was published. I was right, and DL Pharmaceuticals eventually produced it in limited quantities in 2007, only to disappear again by 2008. Recently, Geneza Pharmaceuticals has put it back on the market, as a 50mg tablet. I can understand why they’d think it would be appealing to anabolic steroid users - it’s 3x as androgenic as testosterone and almost 6x as anabolic! While I realize that those numbers don’t always paint an accurate picture of a steroid’s potency (Halotestin is over 19x as anabolic as testosterone, and it’s virtually useless for muscle gain). (*Note: I don’t work for Geneza Pharmaceuticals, aka Naps/NapsGear, nor any of their competitors.)
Taking a look at the metabolites, none are immediately aromatized into estrogen, but what I’m seeing here is a removal of the 4-5 double bond and the addition of a hydrogen, thereby showing the potential of this steroid to become 5a-reduced version of its former self, or a dihydrodimethyltestosterone. Last time I checked, William Llewellyn had been saying that Bolasterone probably wasn’t able to be 5a-reduced, and likely converts to a highly potent estrogen, but I think the chart on the left clearly shows the opposite. I mention this because even though I think he’s a complete D-Bag, I don’t discount his steroid knowledge. None of the metabolites appear to be aromatized, as the signature alternating double bonds in the A-ring are not apparent at this stage. Is there further metabolism of these metabolites downstream? Are they substrates for something I haven’t examined? I don’t know. Maybe there is. Maybe they are. I have no idea.
Methyltestosterone happens to convert to a very potent form of estrogen, so this might be the case here as well, and Bolasterone may well end up being the kind of stuff we see people finding use to necessarily be in conjunction with an anti-estrogen, like Anastrozole (Arimidex) or Aromasin (Exemestane). Maybe it converts to the frightening 7α,17α-dimethylestradiol. And since Cheque drops are a liver-toxic nightmare, in terms of estrogen-like symptoms, we may see that here too…perhaps similarly to what is seen with Anadrol, which is 5a-reduced and doesn’t convert to estrogen – yet for some reason exhibits estrogen like side effects such as gynecomastia. Hell…maybe we won’t see any conversion to anything, and a ton of side effects anyway (again, Anadrol comes to mind). On the other hand, this stuff is definitely going to be liver toxic. But as for side effects? We may see none.
Then again, perhaps is doesn’t convert to estrogen at all. If Bolasterone undergoes 5a-reduction immediately in the first stage of metabolism, then aromatization would be impossible. On the other hand, if this chart is incomplete, then maybe it does undergo conversion to estrogen.
One thing is for sure: Since Geneza Pharmaceuticals has brought this stuff back into circulation, we’ll find out soon enough.
--------------------------------------------------------------------------------------------
Bolasterone is an oral anabolic steroid which is structurally related to methyltestosterone. It differs only by the addition of a methyl group, which is the reasoning for its chemical name. The addition of this methyl group makes the activity of this steroid far different than its cousin however, and makes any comparison between the two difficult. This drug was first developed in the late 1950’s. It was closely evaluated for anabolic and androgenic effect around 3 years later. The drug was developed by the pharmaceutical company UpJohn, and was sold in the United States during the 1960s under the brand name of Myagen. It was mainly prescribed for the treatment of advanced breast cancer in women, but was also investigated for use on lean tissue sparing activity. The medical use of this drug didn’t last long however, and it soon disappeared off the market not too long after it was released. By the 1980s, the drug had pretty much been forgotten by bodybuilders and athletes. Although bolasterone is no longer produced, the drug remains listed in the U.S Pharmacopeias, suggesting that it wouldn’t be impossible to see the drug available once again as a prescription medication in the U.S, however this remains very unlikely.
Bolasterone is a fairly potent anabolic steroid, measured in human subjects to have approximately twice the anabolic effect of methandrostenolone. Despite being a derivative of testosterone, bolasterone is considerably more anabolic than it is androgenic in nature. Bodybuilders and athletes would often use this drug in bulking cycle, where adding extra weight wasn’t a concern. Bolasterone is a very estrogenic steroid by nature, and one can expect to see all of the common estrogen related side effects when taking this drug, especially in higher doses. Estrogen related side effects can include such things as increased water and fat retention and gyno (the development of unattractive and sometimes painful female breast tissue under the nipples in males). To combat such issues, users often prefer to run some sort of anti estrogen compound such as arimidex or aromasin during cycle. This steroid can also be androgenic and can produce androgen related side effects as well. These side effects can include such things as oily skin, acne, and increased body and facial hair. In women, androgen can cause masculizing side effects such as deepening of the voice, the growth facial hair, and clitoral enlargement. Bolasterone is a C17aa compound, which means that it can be toxic to liver if taken in doses too large or for periods too long. Because of this, users are urged to try to keep cycles under 8 weeks and to run some sort of liver protection product such as liv-52. Like all anabolic steroids, bolasterone will shut down the body’s natural testosterone production, making a post cycle therapy protocol necessary after the drug’s use has been discontinued. Users often choose to run compounds such as clomid and HCG to get the body to start producing testosterone naturally again.
Clinical studies have demonstrated that significant nitrogen retention and weight gain can be induced with a daily dosage of 1-2mg per day. In the case of bodybuilders and athletes looking for performance enhancement purposes, users often choose run a dosage of 2-5mg per day for a period of 6-8 weeks. This level is sufficient for strong increases in muscle size and strength, although such gains will likely be accompanied by significant water retention due to estrogen. Bolasterone is generally not recommended for women due to its very strong nature and tendacy to produce virilizing side effects.
MY NOTES CONTINUE PLEASE READ ON
I'll be back later on tonight to update this page with a flood of information and items to think about regarding this supplement.However in the meantime I will simply leave this sexy piece of eye candy here for all to enjoy.
MY NOTES CONTINUE PLEASE READ ON
